Optimization of activity, selectivity, and liability profiles in 5-oxopyrrolopyridine DPP4 inhibitors leading to clinical candidate (Sa)-2-(3-(aminomethyl)-4-(2,4-dichlorophenyl)-2-methyl-5-oxo-5H-pyrrolo[3,4-b]pyridin-6(7H)-yl)-N,N-dimethylacetamide (BMS-767778). [electronic resource]

By: Contributor(s): Producer: 20131126Description: 7343-57 p. digitalISSN:
  • 1520-4804
Subject(s): Online resources: In: Journal of medicinal chemistry vol. 56
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Publication Type: Journal Article

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