Revertants, low temperature, and correctors reveal the mechanism of F508del-CFTR rescue by VX-809 and suggest multiple agents for full correction. [electronic resource]
Producer: 20140623Description: 943-55 p. digitalISSN:- 1879-1301
- Aminopyridines -- pharmacology
- Benzodioxoles -- pharmacology
- Cystic Fibrosis Transmembrane Conductance Regulator -- chemistry
- Drug Synergism
- Endoplasmic Reticulum -- drug effects
- Humans
- Kinetics
- Models, Molecular
- Nucleotides -- metabolism
- Protein Folding -- drug effects
- Protein Structure, Tertiary
- Sequence Deletion -- drug effects
- Temperature
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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