Discovery, synthesis, and structure-activity relationships of 2-aminoquinazoline derivatives as a novel class of metabotropic glutamate receptor 5 negative allosteric modulators. [electronic resource]
Producer: 20140130Description: 4493-500 p. digitalISSN:- 1464-3405
- Allosteric Regulation -- drug effects
- Animals
- Cells, Cultured
- Drug Discovery
- Drug Evaluation, Preclinical
- Humans
- Inhibitory Concentration 50
- Models, Molecular
- Quinazolines -- chemical synthesis
- Quinazolinones -- chemistry
- Rats
- Receptor, Metabotropic Glutamate 5 -- agonists
- Receptors, Metabotropic Glutamate -- agonists
- Structure-Activity Relationship
- Toluidines -- chemistry
- User-Computer Interface
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Publication Type: Journal Article
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