P-glycoprotein (MDR1/ABCB1) and breast cancer resistance protein (BCRP/ABCG2) restrict brain accumulation of the JAK1/2 inhibitor, CYT387. [electronic resource]
Producer: 20140416Description: 9-16 p. digitalISSN:- 1096-1186
- ATP Binding Cassette Transporter, Subfamily B -- genetics
- ATP Binding Cassette Transporter, Subfamily B, Member 1 -- metabolism
- ATP Binding Cassette Transporter, Subfamily G, Member 2
- ATP-Binding Cassette Transporters -- genetics
- Animals
- Benzamides -- blood
- Brain -- metabolism
- Cell Line
- Female
- Gene Deletion
- Humans
- Janus Kinase 1 -- antagonists & inhibitors
- Janus Kinase 2 -- antagonists & inhibitors
- Janus Kinases -- antagonists & inhibitors
- Mice
- Neoplasm Proteins -- metabolism
- Pyrimidines -- blood
- ATP-Binding Cassette Sub-Family B Member 4
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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