Structure-activity relationship study reveals ML240 and ML241 as potent and selective inhibitors of p97 ATPase. [electronic resource]
Producer: 20130703Description: 297-312 p. digitalISSN:- 1860-7187
- Adenosine Triphosphatases -- antagonists & inhibitors
- Antineoplastic Agents -- chemistry
- Autophagy -- drug effects
- Benzimidazoles -- chemistry
- Benzoxazines
- Caspases -- metabolism
- Cell Line, Tumor
- Cell Proliferation -- drug effects
- Endoplasmic Reticulum-Associated Degradation -- drug effects
- Humans
- Neoplasms -- drug therapy
- Nuclear Proteins -- antagonists & inhibitors
- Proteasome Endopeptidase Complex -- metabolism
- Proteasome Inhibitors -- pharmacology
- Quinazolines -- chemistry
- Structure-Activity Relationship
- Ubiquitin -- metabolism
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
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