An optimized RAD51 inhibitor that disrupts homologous recombination without requiring Michael acceptor reactivity. [electronic resource]
Producer: 20130417Description: 254-63 p. digitalISSN:- 1520-4804
- Binding Sites
- DNA -- chemistry
- DNA Repair -- drug effects
- HEK293 Cells
- Homologous Recombination -- drug effects
- Humans
- Maleimides -- chemical synthesis
- Morpholines -- chemical synthesis
- Protein Binding
- Pyrroles -- chemistry
- Rad51 Recombinase -- antagonists & inhibitors
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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