A metal-based inhibitor of NEDD8-activating enzyme. [electronic resource]
Producer: 20130522Description: e49574 p. digitalISSN:- 1932-6203
- Caco-2 Cells
- Cell Line, Tumor
- Cell-Free System
- Cyclopentanes -- pharmacology
- DNA-Binding Proteins -- chemistry
- Dimerization
- Dose-Response Relationship, Drug
- Humans
- Inhibitory Concentration 50
- Ligands
- Luciferases -- metabolism
- Magnetic Resonance Spectroscopy -- methods
- Metals -- chemistry
- Models, Chemical
- Molecular Conformation
- NEDD8 Protein
- NF-kappa B -- metabolism
- Protein Binding
- Pyridines -- chemistry
- Pyrimidines -- pharmacology
- Rhodium -- chemistry
- Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization
- Ubiquitin-Activating Enzymes
- Ubiquitins -- chemistry
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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