Co-crystalization and in vitro biological characterization of 5-aryl-4-(5-substituted-2-4-dihydroxyphenyl)-1,2,3-thiadiazole Hsp90 inhibitors. [electronic resource]
Producer: 20130312Description: e44642 p. digitalISSN:- 1932-6203
- Antineoplastic Agents -- pharmacology
- Apoptosis
- Biomarkers, Tumor -- metabolism
- Cell Line, Tumor
- Crystallization
- Crystallography, X-Ray -- methods
- Drug Screening Assays, Antitumor
- HSP27 Heat-Shock Proteins -- chemistry
- HSP72 Heat-Shock Proteins -- chemistry
- HSP90 Heat-Shock Proteins -- antagonists & inhibitors
- Humans
- In Vitro Techniques
- Inhibitory Concentration 50
- Models, Chemical
- Mutation
- Protein Binding
- Protein Structure, Tertiary
- Recombinant Proteins -- chemistry
- Thiadiazoles -- chemistry
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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