Identification of a new specific Kv1.3 channel blocker, Ctri9577, from the scorpion Chaerilus tricostatus. [electronic resource]
Producer: 20121009Description: 94-9 p. digitalISSN:- 1873-5169
- Amino Acid Sequence
- Animals
- Base Sequence
- Cloning, Molecular
- Dose-Response Relationship, Drug
- HEK293 Cells
- Humans
- Kv1.3 Potassium Channel -- antagonists & inhibitors
- Membrane Potentials -- drug effects
- Models, Molecular
- Molecular Sequence Data
- Molecular Weight
- Patch-Clamp Techniques
- Phylogeny
- Potassium Channel Blockers -- isolation & purification
- Protein Structure, Tertiary
- RNA, Transfer, Amino Acyl
- Recombinant Proteins -- biosynthesis
- Scorpion Venoms -- biosynthesis
- Scorpions -- genetics
- Sequence Analysis, DNA
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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