Oncogenic mutations counteract intrinsic disorder in the EGFR kinase and promote receptor dimerization. [electronic resource]
Producer: 20120702Description: 860-70 p. digitalISSN:- 1097-4172
- Amino Acid Sequence
- Crystallography, X-Ray
- ErbB Receptors -- antagonists & inhibitors
- Gefitinib
- Humans
- Lapatinib
- Molecular Dynamics Simulation
- Molecular Sequence Data
- Neoplasms -- metabolism
- Point Mutation
- Protein Folding
- Protein Kinase Inhibitors -- pharmacology
- Protein Multimerization
- Protein Structure, Tertiary
- Quinazolines -- pharmacology
- Sequence Alignment
- Signal Transduction
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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