Role of human CYP3A4 in the biotransformation of sorafenib to its major oxidized metabolites. [electronic resource]
Producer: 20120809Description: 215-23 p. digitalISSN:- 1873-2968
- Benzenesulfonates -- metabolism
- Catalytic Domain
- Cytochrome P-450 CYP3A -- chemistry
- Humans
- Inactivation, Metabolic
- Microsomes, Liver -- drug effects
- Models, Molecular
- Niacinamide -- analogs & derivatives
- Oxidation-Reduction
- Phenylurea Compounds
- Protein Conformation
- Pyridines -- metabolism
- Sorafenib
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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