The dopaminergic stabilizer pridopidine is to a major extent N-depropylated by CYP2D6 in humans. [electronic resource]
Producer: 20121226Description: 1281-6 p. digitalISSN:- 1432-1041
- Administration, Oral
- Adult
- Area Under Curve
- Biotransformation
- Cytochrome P-450 CYP2D6 -- metabolism
- Cytochrome P-450 CYP2D6 Inhibitors
- Dealkylation
- Dopamine Antagonists -- administration & dosage
- Enzyme Inhibitors -- pharmacokinetics
- Glomerular Filtration Rate
- Half-Life
- Humans
- Intestinal Absorption
- Kidney -- metabolism
- Metabolic Clearance Rate
- Middle Aged
- Phenotype
- Piperidines -- administration & dosage
- Sweden
- White People
- Young Adult
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Publication Type: Clinical Trial; Journal Article; Research Support, Non-U.S. Gov't
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