Saquinavir inhibits the malaria parasite's chloroquine resistance transporter. [electronic resource]
Producer: 20120817Description: 2283-9 p. digitalISSN:- 1098-6596
- Animals
- Antimalarials -- pharmacology
- Biological Transport -- drug effects
- Chloroquine -- pharmacology
- Drug Combinations
- Drug Synergism
- Female
- HIV Protease Inhibitors -- pharmacology
- Humans
- Lopinavir -- pharmacology
- Malaria, Falciparum -- drug therapy
- Membrane Transport Proteins -- genetics
- Mutation
- Oocytes -- cytology
- Plasmodium falciparum -- drug effects
- Protozoan Proteins -- antagonists & inhibitors
- Ritonavir -- pharmacology
- Saquinavir -- pharmacology
- Tritium
- Xenopus laevis
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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