Drug metabolism by CYP2C8.3 is determined by substrate dependent interactions with cytochrome P450 reductase and cytochrome b5. [electronic resource]
Producer: 20111003Description: 681-91 p. digitalISSN:- 1873-2968
- Amino Acid Sequence
- Animals
- Aryl Hydrocarbon Hydroxylases -- genetics
- Catalysis
- Cytochrome P-450 CYP2C8
- Cytochromes b5 -- genetics
- Escherichia coli -- enzymology
- Humans
- In Vitro Techniques
- Inactivation, Metabolic
- Kinetics
- Microsomes, Liver -- drug effects
- Models, Molecular
- Molecular Sequence Data
- NADPH-Ferrihemoprotein Reductase -- genetics
- Oxidation-Reduction
- Pharmaceutical Preparations -- metabolism
- Polymorphism, Genetic
- Protein Binding
- Rats
- Recombinant Proteins -- genetics
- Sequence Alignment
- Substrate Specificity
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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