A series of structurally simple chloroquine chemosensitizing dibemethin derivatives that inhibit chloroquine transport by PfCRT. [electronic resource]
Producer: 20110808Description: 1729-42 p. digitalISSN:- 1768-3254
- Animals
- Antimalarials -- chemical synthesis
- Chloroquine -- antagonists & inhibitors
- Dose-Response Relationship, Drug
- Membrane Transport Proteins -- metabolism
- Methylamines -- chemical synthesis
- Molecular Structure
- Oocytes -- metabolism
- Plasmodium falciparum -- drug effects
- Protozoan Proteins -- metabolism
- Quantitative Structure-Activity Relationship
- Stereoisomerism
- Structure-Activity Relationship
- Xenopus laevis -- metabolism
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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