Design and synthesis of an orally active metabotropic glutamate receptor subtype-2 (mGluR2) positive allosteric modulator (PAM) that decreases cocaine self-administration in rats. [electronic resource]
Producer: 20111109Description: 342-53 p. digitalISSN:- 1520-4804
- Administration, Oral
- Allosteric Regulation
- Animals
- Benzothiazoles -- chemical synthesis
- Biological Availability
- Brain -- metabolism
- Chlorobenzoates -- chemical synthesis
- Cocaine -- administration & dosage
- Cocaine-Related Disorders -- drug therapy
- Drug Design
- HEK293 Cells
- Humans
- Rats
- Receptors, Metabotropic Glutamate -- physiology
- Self Administration
- Structure-Activity Relationship
- Tissue Distribution
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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