Dipeptidyl-quinolone derivatives inhibit hypoxia inducible factor-1α prolyl hydroxylases-1, -2, and -3 with altered selectivity. [electronic resource]
Producer: 20101223Description: 676-86 p. digitalISSN:- 1520-4774
- Combinatorial Chemistry Techniques
- Dipeptides -- chemical synthesis
- Enzyme Inhibitors -- chemical synthesis
- Hypoxia-Inducible Factor 1, alpha Subunit -- metabolism
- Isoenzymes -- antagonists & inhibitors
- Molecular Structure
- Procollagen-Proline Dioxygenase -- antagonists & inhibitors
- Quinolones -- chemical synthesis
- Stereoisomerism
- Structure-Activity Relationship
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Publication Type: Journal Article
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