Metabolism of fostamatinib, the oral methylene phosphate prodrug of the spleen tyrosine kinase inhibitor R406 in humans: contribution of hepatic and gut bacterial processes to the overall biotransformation. [electronic resource]
Producer: 20101012Description: 1166-76 p. digitalISSN:- 1521-009X
- Adult
- Aminopyridines
- Bacteria, Anaerobic -- metabolism
- Biotransformation
- Gastrointestinal Tract -- metabolism
- Humans
- In Vitro Techniques
- Inactivation, Metabolic
- Liver -- metabolism
- Male
- Microsomes -- metabolism
- Morpholines
- Oxazines -- pharmacokinetics
- Prodrugs -- pharmacokinetics
- Pyridines -- pharmacokinetics
- Pyrimidines
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Publication Type: Journal Article
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