Function of activation loop tyrosine phosphorylation in the mechanism of c-Kit auto-activation and its implication in sunitinib resistance. [electronic resource]
Producer: 20100716Description: 601-9 p. digitalISSN:- 1756-2651
- Amino Acid Substitution
- Antineoplastic Agents -- metabolism
- Benzamides
- Catalytic Domain
- Drug Resistance, Neoplasm
- Enzyme Activation
- Enzyme Inhibitors -- metabolism
- Humans
- Imatinib Mesylate
- Indoles -- metabolism
- Kinetics
- Microchemistry -- methods
- Models, Biological
- Mutant Proteins -- chemistry
- Peptide Mapping
- Phosphorylation
- Phosphotyrosine -- physiology
- Piperazines -- metabolism
- Protein Binding
- Protein Interaction Domains and Motifs -- physiology
- Proto-Oncogene Proteins c-kit -- antagonists & inhibitors
- Pyrimidines -- metabolism
- Pyrroles -- metabolism
- Recombinant Fusion Proteins -- antagonists & inhibitors
- Sunitinib
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Publication Type: Journal Article
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