Screening for antibacterial inhibitors of the UDP-3-O-(R-3-hydroxymyristoyl)-N-acetylglucosamine deacetylase (LpxC) using a high-throughput mass spectrometry assay. [electronic resource]
Producer: 20100318Description: 52-61 p. digitalISSN:- 1552-454X
- Amidohydrolases -- antagonists & inhibitors
- Anti-Bacterial Agents -- analysis
- Dimethyl Sulfoxide -- pharmacology
- Enzyme Inhibitors -- analysis
- Enzyme Stability -- drug effects
- Escherichia coli -- drug effects
- Fluorescence
- High-Throughput Screening Assays -- methods
- Mass Spectrometry -- methods
- Microbial Sensitivity Tests
- Reproducibility of Results
- Small Molecule Libraries -- analysis
- Substrate Specificity -- drug effects
- Temperature
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Publication Type: Journal Article
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