An NSAID-like compound, FT-9, preferentially inhibits gamma-secretase cleavage of the amyloid precursor protein compared to its effect on amyloid precursor-like protein 1. [electronic resource]
Producer: 20091231Description: 10894-904 p. digitalISSN:- 1520-4995
- Amyloid Precursor Protein Secretases -- antagonists & inhibitors
- Amyloid beta-Peptides -- metabolism
- Amyloid beta-Protein Precursor -- metabolism
- Animals
- Anti-Inflammatory Agents, Non-Steroidal -- pharmacology
- Benzodiazepinones -- pharmacology
- Biocatalysis -- drug effects
- CHO Cells
- Cricetinae
- Cricetulus
- Dipeptides -- pharmacology
- Fenofibrate -- analogs & derivatives
- Flurbiprofen -- pharmacology
- Humans
- Kinetics
- Microsomes -- drug effects
- Nerve Tissue Proteins -- metabolism
- Peptide Fragments -- metabolism
- Protease Inhibitors -- pharmacology
- Recombinant Proteins -- genetics
- Substrate Specificity -- drug effects
- Transfection
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
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