Silencing the cochaperone CDC37 destabilizes kinase clients and sensitizes cancer cells to HSP90 inhibitors. [electronic resource]
Producer: 20090507Description: 157-69 p. digitalISSN:- 1476-5594
- Adenocarcinoma -- metabolism
- Apoptosis -- drug effects
- Benzoquinones -- pharmacology
- Breast Neoplasms -- metabolism
- Cell Cycle Proteins -- antagonists & inhibitors
- Cell Division -- drug effects
- Cell Line, Tumor -- drug effects
- Chaperonins -- antagonists & inhibitors
- Colonic Neoplasms -- metabolism
- Female
- G1 Phase -- drug effects
- Gene Expression Regulation, Neoplastic -- drug effects
- Gene Targeting
- HSP90 Heat-Shock Proteins -- antagonists & inhibitors
- Humans
- Lactams, Macrocyclic -- pharmacology
- Male
- Neoplasm Proteins -- antagonists & inhibitors
- Phosphorylation -- drug effects
- Prostatic Neoplasms -- metabolism
- Proteasome Endopeptidase Complex -- metabolism
- Protein Kinases -- metabolism
- Protein Processing, Post-Translational -- drug effects
- Pyrazoles -- pharmacology
- RNA Interference
- RNA, Small Interfering -- pharmacology
- Signal Transduction -- drug effects
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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