Significant antitumor activity in vivo following treatment with the microtubule agent ENMD-1198. [electronic resource]
Producer: 20080822Description: 1472-82 p. digitalISSN:- 1535-7163
- 2-Methoxyestradiol
- Administration, Oral
- Animals
- Antineoplastic Agents -- administration & dosage
- Apoptosis -- drug effects
- Binding, Competitive -- drug effects
- Cell Line, Tumor
- Cell Proliferation -- drug effects
- Colchicine -- pharmacology
- Drug Screening Assays, Antitumor
- Estradiol -- analogs & derivatives
- Estrenes -- administration & dosage
- G2 Phase -- drug effects
- Hepatocytes -- drug effects
- Humans
- Hypoxia-Inducible Factor 1, alpha Subunit -- metabolism
- Inhibitory Concentration 50
- Male
- Mice
- Mice, Inbred C57BL
- Microtubules -- drug effects
- Mitosis -- drug effects
- Rats
- Survival Analysis
- Tubulin -- metabolism
- Tubulin Modulators -- administration & dosage
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Publication Type: Journal Article
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