Rational design of novel, potent piperazinone and imidazolidinone BACE1 inhibitors. [electronic resource]
Producer: 20080709Description: 3236-41 p. digitalISSN:- 1464-3405
- Amyloid Precursor Protein Secretases -- antagonists & inhibitors
- Animals
- Aspartic Acid Endopeptidases -- antagonists & inhibitors
- Crystallography, X-Ray
- Disease Models, Animal
- Drug Design
- Humans
- Imidazolidines -- chemical synthesis
- Mice
- Mice, Transgenic
- Models, Molecular
- Molecular Conformation
- Molecular Structure
- Piperazines -- chemical synthesis
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, U.S. Gov't, Non-P.H.S.
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