Small-molecule screen identifies inhibitors of a human intestinal calcium-activated chloride channel. [electronic resource]
Producer: 20080407Description: 758-68 p. digitalISSN:- 1521-0111
- Adenosine Triphosphate -- antagonists & inhibitors
- Calcium -- analysis
- Carbachol -- antagonists & inhibitors
- Chloride Channels -- antagonists & inhibitors
- Chlorides -- metabolism
- Dose-Response Relationship, Drug
- Drug Evaluation, Preclinical -- methods
- Fluorescent Dyes -- metabolism
- Fura-2 -- metabolism
- Genetic Vectors
- HT29 Cells
- Humans
- Inhibitory Concentration 50
- Intestinal Mucosa -- metabolism
- Intestines -- drug effects
- Ion Channel Gating -- drug effects
- Kinetics
- Lentivirus -- genetics
- Models, Biological
- Molecular Structure
- Patch-Clamp Techniques
- Reproducibility of Results
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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