Nonsteroidal glucocorticoid agonists: tetrahydronaphthalenes with alternative steroidal A-ring mimetics possessing dissociated (transrepression/transactivation) efficacy selectivity. [electronic resource]
Producer: 20080403Description: 6519-34 p. digitalISSN:- 0022-2623
- Anti-Inflammatory Agents, Non-Steroidal -- chemical synthesis
- Binding Sites
- Cell Line
- Drug Partial Agonism
- Humans
- Mammary Tumor Virus, Mouse -- genetics
- Models, Molecular
- Molecular Mimicry
- NF-kappa B -- genetics
- Receptors, Glucocorticoid -- agonists
- Stereoisomerism
- Structure-Activity Relationship
- Tetrahydronaphthalenes -- chemical synthesis
- Transcription, Genetic -- drug effects
- Transcriptional Activation -- drug effects
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Publication Type: Journal Article
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