Identification of human liver cytochrome P450 enzymes involved in biotransformation of vicriviroc, a CCR5 receptor antagonist. [electronic resource]
Producer: 20080103Description: 2186-95 p. digitalISSN:- 0090-9556
- Antibodies, Monoclonal
- Aryl Hydrocarbon Hydroxylases -- metabolism
- Biotransformation
- Bridged-Ring Compounds -- pharmacology
- CCR5 Receptor Antagonists
- Carboxylic Acids -- metabolism
- Cytochrome P-450 CYP2C9
- Cytochrome P-450 CYP3A
- Cytochrome P-450 Enzyme Inhibitors
- Cytochrome P-450 Enzyme System -- immunology
- Dealkylation
- Enzyme Inhibitors -- pharmacology
- Humans
- Immunologic Factors -- metabolism
- In Vitro Techniques
- Isoenzymes -- metabolism
- Ketoconazole -- pharmacology
- Kinetics
- Liver -- drug effects
- Oxidation-Reduction
- Piperazines -- metabolism
- Pyrimidines -- metabolism
- Recombinant Proteins -- metabolism
- Substrate Specificity
- Testosterone -- metabolism
- Triazoles -- pharmacology
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Publication Type: Journal Article
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