Multiple human isoforms of drug transporters contribute to the hepatic and renal transport of olmesartan, a selective antagonist of the angiotensin II AT1-receptor. [electronic resource]
Producer: 20080103Description: 2166-76 p. digitalISSN:- 0090-9556
- ATP Binding Cassette Transporter, Subfamily B
- ATP Binding Cassette Transporter, Subfamily B, Member 1 -- metabolism
- ATP Binding Cassette Transporter, Subfamily G, Member 2
- ATP-Binding Cassette Transporters -- metabolism
- Adenosine Triphosphate -- metabolism
- Angiotensin II Type 1 Receptor Blockers -- metabolism
- Animals
- Cell Line
- Dogs
- Dose-Response Relationship, Drug
- Estrone -- analogs & derivatives
- Female
- Hepatocytes -- drug effects
- Humans
- Imidazoles -- metabolism
- In Vitro Techniques
- Kidney -- metabolism
- Kinetics
- Liver -- drug effects
- Liver-Specific Organic Anion Transporter 1
- Membrane Transport Proteins -- drug effects
- Mice
- Mice, Knockout
- Multidrug Resistance-Associated Protein 2
- Multidrug Resistance-Associated Proteins -- deficiency
- Neoplasm Proteins -- metabolism
- Olmesartan Medoxomil
- Organic Anion Transporters -- metabolism
- Organic Anion Transporters, Sodium-Independent -- metabolism
- Penicillin G -- pharmacology
- Probenecid -- pharmacology
- Prodrugs -- metabolism
- Protein Binding
- Protein Isoforms -- metabolism
- Sincalide -- metabolism
- Solute Carrier Organic Anion Transporter Family Member 1B3
- Tetrazoles -- metabolism
- Transfection
- p-Aminohippuric Acid -- pharmacology
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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