Farnesyl transferase inhibitors impair chromosomal maintenance in cell lines and human tumors by compromising CENP-E and CENP-F function. [electronic resource]
Producer: 20070612Description: 1317-28 p. digitalISSN:- 1535-7163
- Binding Sites -- drug effects
- Cell Line, Tumor
- Cell Proliferation -- drug effects
- Chromosomal Proteins, Non-Histone -- metabolism
- Chromosomes, Human -- drug effects
- Enzyme Activation -- drug effects
- Enzyme Inhibitors -- chemistry
- Farnesyltranstransferase -- antagonists & inhibitors
- Head and Neck Neoplasms -- drug therapy
- Humans
- Kinetochores -- drug effects
- Metaphase -- drug effects
- Microfilament Proteins -- metabolism
- Microtubules -- drug effects
- Piperidines -- chemistry
- Prometaphase -- drug effects
- Protein Kinases -- metabolism
- Protein Serine-Threonine Kinases
- Pyridines -- chemistry
- Spindle Apparatus -- drug effects
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Publication Type: Clinical Trial, Phase I; Journal Article; Randomized Controlled Trial; Research Support, N.I.H., Extramural
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