Amodiaquine metabolism is impaired by common polymorphisms in CYP2C8: implications for malaria treatment in Africa. [electronic resource]
Producer: 20070911Description: 197-203 p. digitalISSN:- 0009-9236
- Alkynes
- Amodiaquine -- analogs & derivatives
- Antimalarials -- metabolism
- Aryl Hydrocarbon Hydroxylases -- genetics
- Benzoxazines -- metabolism
- Burkina Faso
- Chromatography, High Pressure Liquid
- Cyclopropanes
- Cytochrome P-450 CYP2C8
- Dose-Response Relationship, Drug
- Drug Interactions
- Enzyme Inhibitors -- metabolism
- Genotype
- HIV Protease Inhibitors -- metabolism
- Humans
- Lopinavir
- Malaria, Falciparum -- drug therapy
- Models, Biological
- Polymorphism, Genetic
- Pyridines -- metabolism
- Pyrimidinones -- metabolism
- Pyrones -- metabolism
- Reverse Transcriptase Inhibitors -- metabolism
- Saquinavir -- metabolism
- Spectrophotometry, Ultraviolet
- Sulfonamides
- Treatment Outcome
- Trimethoprim -- metabolism
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, N.I.H., Intramural
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