Methyl succinate antagonises biguanide-induced AMPK-activation and death of pancreatic beta-cells through restoration of mitochondrial electron transfer. [electronic resource]
Producer: 20070524Description: 1031-43 p. digitalISSN:- 0007-1188
- AMP-Activated Protein Kinases
- Animals
- Apoptosis -- drug effects
- Biguanides -- antagonists & inhibitors
- Cell Line, Tumor
- Cell Survival -- drug effects
- Dose-Response Relationship, Drug
- Electron Transport -- drug effects
- Electron Transport Complex I -- antagonists & inhibitors
- Electron Transport Complex II -- drug effects
- Enzyme Activation -- drug effects
- Glucose -- metabolism
- Hypoglycemic Agents -- antagonists & inhibitors
- Insulin-Secreting Cells -- drug effects
- Metformin -- toxicity
- Mice
- Mitochondria -- drug effects
- Multienzyme Complexes -- metabolism
- NADP -- metabolism
- Oxidation-Reduction
- Phenformin -- toxicity
- Phosphorylation -- drug effects
- Protein Serine-Threonine Kinases -- metabolism
- Rats
- Succinates -- metabolism
- Tetrazolium Salts -- metabolism
- Thiazoles -- metabolism
- Time Factors
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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