Small-molecule inhibition of the interaction between the translation initiation factors eIF4E and eIF4G. [electronic resource]
Producer: 20070313Description: 257-67 p. digitalISSN:- 0092-8674
- Animals
- Antineoplastic Agents -- chemistry
- Cell Line, Transformed
- Cell Line, Tumor
- Cell Transformation, Neoplastic -- drug effects
- Drug Evaluation, Preclinical -- methods
- Eukaryotic Initiation Factor-4E -- drug effects
- Eukaryotic Initiation Factor-4G -- drug effects
- Feedback, Physiological -- drug effects
- Fluorescence Polarization Immunoassay -- methods
- Gene Expression Regulation, Neoplastic -- drug effects
- Humans
- Hydrazones
- Jurkat Cells
- Mice
- Models, Molecular
- Nitro Compounds -- chemistry
- Oncogenes -- drug effects
- Peptide Fragments -- genetics
- Protein Binding -- drug effects
- Protein Biosynthesis -- drug effects
- RNA, Messenger -- drug effects
- Thiazoles -- chemistry
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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