Topographical requirements for delta opioid ligands: presence of a carboxyl group in position 4 is not critical for deltorphin high delta receptor affinity and analgesic activity. [electronic resource]
Producer: 19911216Description: 1290-7 p. digitalISSN:- 0006-291X
- Amino Acid Sequence
- Analgesics -- chemistry
- Animals
- Binding, Competitive
- Brain -- metabolism
- Male
- Models, Molecular
- Molecular Sequence Data
- Oligopeptides -- chemical synthesis
- Pain
- Protein Conformation
- Radioligand Assay
- Rats
- Rats, Inbred Strains
- Receptors, Opioid -- drug effects
- Receptors, Opioid, delta
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Publication Type: Comparative Study; Journal Article; Research Support, U.S. Gov't, P.H.S.
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