Structural determinants of Torpedo californica acetylcholinesterase inhibition by the novel and orally active carbamate based anti-alzheimer drug ganstigmine (CHF-2819). [electronic resource]
Producer: 20061003Description: 5051-8 p. digitalISSN:- 0022-2623
- Acetylcholinesterase -- chemistry
- Administration, Oral
- Alkaloids -- administration & dosage
- Alzheimer Disease -- drug therapy
- Animals
- Binding Sites -- drug effects
- Brain -- enzymology
- Carbamates -- administration & dosage
- Cholinesterase Inhibitors -- administration & dosage
- Crystallization
- Crystallography, X-Ray
- Drug Evaluation, Preclinical
- Enzyme Activation -- drug effects
- Male
- Mice
- Models, Molecular
- Molecular Conformation
- Stereoisomerism
- Structure-Activity Relationship
- Torpedo
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Publication Type: Comparative Study; Journal Article
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