Pioglitazone is metabolised by CYP2C8 and CYP3A4 in vitro: potential for interactions with CYP2C8 inhibitors. [electronic resource]
Producer: 20061208Description: 44-51 p. digitalISSN:- 1742-7835
- Aryl Hydrocarbon Hydroxylases -- antagonists & inhibitors
- Cytochrome P-450 CYP2C8
- Cytochrome P-450 CYP3A
- Cytochrome P-450 Enzyme System -- metabolism
- Drug Interactions
- Enzyme Inhibitors -- pharmacology
- Humans
- Hypoglycemic Agents -- pharmacokinetics
- In Vitro Techniques
- Microsomes, Liver -- drug effects
- NADP -- metabolism
- Pioglitazone
- Thiazolidinediones -- pharmacokinetics
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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