The second generation of BCR-ABL tyrosine kinase inhibitors. [electronic resource]
Producer: 20060718Description: 294-300 p. digitalISSN:- 0925-5710
- Allosteric Regulation -- drug effects
- Antineoplastic Agents -- chemistry
- Binding Sites -- drug effects
- Drug Design
- Drug Resistance, Neoplasm -- drug effects
- Fusion Proteins, bcr-abl
- Gene Amplification -- drug effects
- Gene Expression Regulation, Leukemic -- drug effects
- Humans
- Leukemia, Myelogenous, Chronic, BCR-ABL Positive -- drug therapy
- Mutation
- Philadelphia Chromosome
- Protein Binding -- drug effects
- Protein Kinase Inhibitors -- chemistry
- Protein Structure, Tertiary -- drug effects
- Protein-Tyrosine Kinases -- antagonists & inhibitors
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Publication Type: Journal Article; Review
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