Telithromycin, but not montelukast, increases the plasma concentrations and effects of the cytochrome P450 3A4 and 2C8 substrate repaglinide. [electronic resource]
Producer: 20060404Description: 231-42 p. digitalISSN:- 0009-9236
- Acetates -- pharmacology
- Adolescent
- Adult
- Area Under Curve
- Aryl Hydrocarbon Hydroxylases -- metabolism
- Biotransformation
- Blood Glucose -- metabolism
- Carbamates -- blood
- Cross-Over Studies
- Cyclopropanes
- Cytochrome P-450 CYP2C8
- Cytochrome P-450 CYP3A
- Cytochrome P-450 Enzyme System -- metabolism
- Drug Interactions
- Female
- Humans
- Hypoglycemic Agents -- blood
- Ketolides -- pharmacology
- Leukotriene Antagonists -- pharmacology
- Male
- Piperidines -- blood
- Quinolines -- pharmacology
- Sulfides
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Publication Type: Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't
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