Dual antagonists of the bradykinin B1 and B2 receptors based on a postulated common pharmacophore from existing non-peptide antagonists. [electronic resource]
Producer: 20060707Description: 189-94 p. digitalISSN:- 1431-6730
- Acetanilides -- chemistry
- Animals
- Aorta -- drug effects
- Binding Sites
- Binding, Competitive
- Bradykinin B1 Receptor Antagonists
- Bradykinin B2 Receptor Antagonists
- Cells, Cultured
- Molecular Structure
- Muscle, Smooth -- chemistry
- Pyrrolidines -- chemistry
- Quinolines -- chemistry
- Quinoxalines -- chemistry
- Rabbits
- Receptor, Bradykinin B1 -- chemistry
- Receptor, Bradykinin B2 -- chemistry
- Structure-Activity Relationship
- Sulfones -- chemistry
- Thiosemicarbazones -- chemistry
- Tosyl Compounds -- chemistry
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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