Tricyclic azepine derivatives: pyrimido[4,5-b]-1,4-benzoxazepines as a novel class of epidermal growth factor receptor kinase inhibitors. [electronic resource]
Producer: 20060417Description: 1643-6 p. digitalISSN:- 0960-894X
- Adenosine Triphosphate -- metabolism
- Azepines -- chemical synthesis
- Binding Sites
- Cell Proliferation -- drug effects
- Cells, Cultured
- ErbB Receptors -- antagonists & inhibitors
- Humans
- Molecular Structure
- Phosphorylation -- drug effects
- Protein Kinase Inhibitors -- chemical synthesis
- Protein Serine-Threonine Kinases -- antagonists & inhibitors
- Protein-Tyrosine Kinases -- antagonists & inhibitors
- Receptor, ErbB-2 -- antagonists & inhibitors
- Structure-Activity Relationship
- Substrate Specificity
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Publication Type: Journal Article
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