[3H]linopirdine binding to rat brain membranes is not relevant for M-channel interaction. [electronic resource]
Producer: 20050923Description: 10-7 p. digitalISSN:- 0014-2999
- Animals
- Anthracenes -- pharmacology
- Binding, Competitive -- drug effects
- Brain -- metabolism
- CHO Cells
- Cell Membrane -- metabolism
- Chlorides -- metabolism
- Cricetinae
- Cricetulus
- Cytochrome P-450 CYP2D6 -- metabolism
- Cytochrome P-450 CYP3A
- Cytochrome P-450 Enzyme System -- metabolism
- Dose-Response Relationship, Drug
- Indoles -- metabolism
- KCNQ3 Potassium Channel
- Ketoconazole -- pharmacology
- Kinetics
- Liver -- metabolism
- Male
- Miconazole -- pharmacology
- Potassium Channels, Voltage-Gated -- antagonists & inhibitors
- Pyridines -- metabolism
- Pyrilamine -- pharmacology
- Quinidine -- pharmacology
- Radioligand Assay
- Rats
- Rats, Sprague-Dawley
- Rubidium -- metabolism
- Tritium
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Publication Type: Comparative Study; Journal Article
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