Drug targeting of HIV-1 RNA.DNA hybrid structures: thermodynamics of recognition and impact on reverse transcriptase-mediated ribonuclease H activity and viral replication. [electronic resource]
Producer: 20040924Description: 9732-42 p. digitalISSN:- 0006-2960
- Aminoglycosides -- pharmacology
- Binding, Competitive
- Circular Dichroism
- DNA, Viral -- antagonists & inhibitors
- Drug Delivery Systems -- methods
- Enzyme Activation -- genetics
- HIV Reverse Transcriptase -- antagonists & inhibitors
- HIV-1 -- drug effects
- Humans
- Hydrolysis -- drug effects
- Neomycin -- metabolism
- Nucleic Acid Conformation
- Nucleic Acid Heteroduplexes -- antagonists & inhibitors
- Paromomycin -- metabolism
- RNA, Viral -- antagonists & inhibitors
- Reverse Transcriptase Inhibitors -- metabolism
- Ribonuclease H -- antagonists & inhibitors
- Ribostamycin -- metabolism
- Thermodynamics
- Virus Replication -- genetics
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Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
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