Sequence-based design of kinase inhibitors applicable for therapeutics and target identification. [electronic resource]
Producer: 20040210Description: 1242-55 p. digitalISSN:- 0021-9258
- 3-Phosphoinositide-Dependent Protein Kinases
- Amino Acid Sequence
- Animals
- Aorta -- metabolism
- Catalytic Domain
- Cell Cycle Proteins -- metabolism
- Cell Division
- Cell Line, Tumor
- Cell-Free System
- Cloning, Molecular
- Cyclin-Dependent Kinase Inhibitor p27
- Cytosol -- metabolism
- DNA Mutational Analysis
- Dose-Response Relationship, Drug
- Drug Design
- Glutathione Transferase -- metabolism
- Humans
- Immunoblotting
- Male
- Mice
- Mice, Inbred BALB C
- Models, Molecular
- Molecular Sequence Data
- Myristic Acids -- metabolism
- Peptides -- chemistry
- Phosphorylation
- Protein Binding
- Protein Serine-Threonine Kinases -- metabolism
- Protein Structure, Tertiary
- Proto-Oncogene Proteins -- metabolism
- Proto-Oncogene Proteins c-akt
- Proto-Oncogene Proteins c-kit -- metabolism
- Substrate Specificity
- Tumor Suppressor Proteins -- metabolism
- src-Family Kinases -- metabolism
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Publication Type: Journal Article
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