Structure-activity relationships of 1-alkyl-5-(3,4-dichlorophenyl)- 5-[2-[(3-substituted)-1-azetidinyl]ethyl]-2-piperidones. 1. Selective antagonists of the neurokinin-2 receptor. [electronic resource]
Producer: 20021220Description: 5365-77 p. digitalISSN:- 0022-2623
- Animals
- Azetidines -- chemical synthesis
- CHO Cells
- Cricetinae
- Drug Stability
- Humans
- In Vitro Techniques
- Microsomes, Liver -- metabolism
- Muscle Contraction -- drug effects
- Muscle, Smooth -- drug effects
- Piperazines -- chemical synthesis
- Piperidones -- chemical synthesis
- Pulmonary Artery -- drug effects
- Rabbits
- Radioligand Assay
- Receptors, Neurokinin-2 -- antagonists & inhibitors
- Receptors, Neurokinin-3 -- metabolism
- Stereoisomerism
- Structure-Activity Relationship
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Publication Type: Journal Article
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