(-)U50,488H [(trans)-3,4-dichloro-N-methyl-N-[2-(1-pyrrolidinyl)-cyclohexyl]benzeneacetamide] induces internalization and down-regulation of the human, but not the rat, kappa-opioid receptor: structural basis for the differential regulation. [electronic resource]
Producer: 20020918Description: 1184-92 p. digitalISSN:- 0022-3565
- 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer -- pharmacology
- Amino Acid Sequence
- Analgesics, Non-Narcotic -- pharmacology
- Animals
- CHO Cells
- Cell Membrane -- metabolism
- Cricetinae
- Diprenorphine -- metabolism
- Down-Regulation -- drug effects
- Fluorescent Antibody Technique, Direct
- Humans
- Intracellular Membranes -- metabolism
- Ionophores -- pharmacology
- Molecular Sequence Data
- Monensin -- pharmacology
- Mutation -- drug effects
- Narcotic Antagonists -- metabolism
- Rats
- Receptors, Opioid, kappa -- biosynthesis
- Recombinant Fusion Proteins -- chemistry
- Species Specificity
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Publication Type: Comparative Study; Journal Article; Research Support, U.S. Gov't, P.H.S.
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