High-affinity activators of cystic fibrosis transmembrane conductance regulator (CFTR) chloride conductance identified by high-throughput screening. [electronic resource]
Producer: 20021120Description: 37235-41 p. digitalISSN:- 0021-9258
- Animals
- Bacterial Proteins -- genetics
- Cells, Cultured
- Colforsin -- pharmacology
- Cystic Fibrosis -- genetics
- Cystic Fibrosis Transmembrane Conductance Regulator -- agonists
- Drug Evaluation, Preclinical -- instrumentation
- Epithelial Cells -- drug effects
- Equipment Design
- Genes, Reporter
- Humans
- Iodides -- pharmacology
- Kinetics
- Luminescent Proteins -- genetics
- Rats
- Rats, Inbred F344
- Recombinant Fusion Proteins -- metabolism
- Respiratory Mucosa -- drug effects
- Structure-Activity Relationship
- Thyroid Gland
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
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