Molecular basis of differences in (-)(trans)-3,4-dichloro-N-methyl-N-[2-(1-pyrrolidiny)-cyclohexyl]benzeneacetamide-induced desensitization and phosphorylation between human and rat kappa-opioid receptors expressed in Chinese hamster ovary cells. [electronic resource]
Producer: 20020110Description: 73-84 p. digitalISSN:- 0026-895X
- 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer -- pharmacology
- Amino Acid Sequence
- Analgesics, Non-Narcotic -- pharmacology
- Animals
- Arrestins -- metabolism
- CHO Cells
- Cricetinae
- Cyclic AMP-Dependent Protein Kinases -- metabolism
- Diprenorphine -- pharmacology
- G-Protein-Coupled Receptor Kinase 3
- Gene Expression -- drug effects
- Guanosine 5'-O-(3-Thiotriphosphate) -- metabolism
- Humans
- Molecular Sequence Data
- Phosphoproteins -- metabolism
- Phosphorylation -- drug effects
- Protein Serine-Threonine Kinases -- metabolism
- Protein Structure, Tertiary
- Rats
- Receptors, Opioid, kappa -- agonists
- Recombinant Fusion Proteins -- drug effects
- Sequence Homology, Amino Acid
- Species Specificity
- Sulfur Radioisotopes
- Transfection
- Tritium
- beta-Adrenergic Receptor Kinases
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Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
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