An interaction between the cytochrome P450 probe substrates chlorzoxazone (CYP2E1) and midazolam (CYP3A). [electronic resource]
Producer: 20020306Description: 555-61 p. digitalISSN:- 0306-5251
- Administration, Oral
- Adult
- Area Under Curve
- Aryl Hydrocarbon Hydroxylases
- Caffeine -- pharmacokinetics
- Chlorzoxazone -- pharmacokinetics
- Cross-Over Studies
- Cytochrome P-450 CYP2E1 -- metabolism
- Cytochrome P-450 CYP3A
- Cytochrome P-450 Enzyme System -- metabolism
- Debrisoquin -- pharmacokinetics
- Diclofenac -- pharmacokinetics
- Drug Interactions
- Female
- Humans
- Male
- Mephenytoin -- pharmacokinetics
- Midazolam -- blood
- Muscle Relaxants, Central -- pharmacokinetics
- Oxidoreductases, N-Demethylating -- metabolism
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Publication Type: Clinical Trial; Journal Article; Randomized Controlled Trial
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