G protein-coupled receptor kinase 2 mediates mu-opioid receptor desensitization in GABAergic neurons of the nucleus raphe magnus. [electronic resource]
Producer: 20010517Description: 435-44 p. digitalISSN:- 0022-3042
- Amino Acid Sequence
- Analgesics, Opioid -- pharmacology
- Animals
- Binding Sites
- Cyclic AMP-Dependent Protein Kinases -- biosynthesis
- Drug Tolerance -- physiology
- Enkephalin, Ala(2)-MePhe(4)-Gly(5)- -- pharmacology
- G-Protein-Coupled Receptor Kinase 2
- G-Protein-Coupled Receptor Kinase 3
- Glutamate Decarboxylase -- biosynthesis
- Ion Transport -- drug effects
- Membrane Potentials -- drug effects
- Molecular Sequence Data
- Nerve Tissue Proteins -- biosynthesis
- Neurons -- drug effects
- Oligopeptides -- chemical synthesis
- Pain -- physiopathology
- Patch-Clamp Techniques
- Phosphorylation
- Potassium -- metabolism
- Potassium Channels -- metabolism
- Potassium Channels, Inwardly Rectifying
- Protein Processing, Post-Translational
- Protein Serine-Threonine Kinases -- biosynthesis
- Protein Structure, Tertiary
- Protein Transport -- drug effects
- RNA, Messenger -- biosynthesis
- Raphe Nuclei -- drug effects
- Rats
- Rats, Sprague-Dawley
- Receptors, Opioid, mu -- agonists
- Reverse Transcriptase Polymerase Chain Reaction
- Signal Transduction -- drug effects
- Spinal Cord -- physiopathology
- beta-Adrenergic Receptor Kinases
- gamma-Aminobutyric Acid -- physiology
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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