Mutation of a single conserved tryptophan in multidrug resistance protein 1 (MRP1/ABCC1) results in loss of drug resistance and selective loss of organic anion transport. [electronic resource]
Producer: 20010614Description: 15616-24 p. digitalISSN:- 0021-9258
- ATP-Binding Cassette Transporters -- chemistry
- Amino Acid Sequence
- Amino Acid Substitution
- Arsenites -- pharmacology
- Binding Sites
- Biological Transport
- Cell Line
- Cell Survival -- drug effects
- Cloning, Molecular
- Conserved Sequence
- Drug Resistance, Multiple
- Genes, Reporter
- Glucuronides -- metabolism
- Green Fluorescent Proteins
- HeLa Cells
- Humans
- Kinetics
- Luminescent Proteins -- genetics
- Molecular Sequence Data
- Multidrug Resistance-Associated Proteins
- Mutagenesis, Site-Directed
- Protein Conformation
- Recombinant Fusion Proteins -- chemistry
- Sequence Alignment
- Sequence Homology, Amino Acid
- Sodium Compounds -- pharmacology
- Transfection
- Tryptophan
- Vincristine -- pharmacokinetics
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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