Amino acid 305 determines catalytic center accessibility in CYP3A4. [electronic resource]
Producer: 20000616Description: 4406-14 p. digitalISSN:- 0006-2960
- Alanine -- genetics
- Amino Acid Substitution -- genetics
- Aryl Hydrocarbon Hydroxylases
- Binding Sites
- Catalysis -- drug effects
- Clotrimazole -- pharmacology
- Cytochrome P-450 CYP3A
- Cytochrome P-450 Enzyme Inhibitors
- Cytochrome P-450 Enzyme System -- chemistry
- Diazepam -- metabolism
- Econazole -- pharmacology
- Erythromycin -- metabolism
- Humans
- Imidazoles -- chemistry
- Ketoconazole -- metabolism
- Kinetics
- Miconazole -- pharmacology
- Mixed Function Oxygenases -- antagonists & inhibitors
- Multienzyme Complexes -- antagonists & inhibitors
- Mutation -- genetics
- Nifedipine -- metabolism
- Oxidoreductases, N-Demethylating -- antagonists & inhibitors
- Substrate Specificity
- Testosterone -- metabolism
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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